Annual Reports Medicinal Chemistry Volume 1 by By C.K. Cain

By By C.K. Cain

Show description

Read or Download Annual Reports Medicinal Chemistry Volume 1 PDF

Similar organic books

Organic Chemistry, Fourth Edition

This leading edge publication from acclaimed educator Paula Bruice is geared up in a fashion that daunts rote memorization. The author's writing has been praised for watching for readers' questions, and appeals to their have to research visually and through fixing difficulties. Emphasizing that newcomers may still cause their technique to strategies instead of memorize proof, Bruice encourages them to contemplate what they've got realized formerly and follow that wisdom in a brand new environment.

Comprehensive Organic Functional Group Transformations, Volume 2 (Synthesis: Carbon with One Heteroatom Attached by a Single Bond)

This quantity describes all tools for the synthesis of compounds containing acarbon atom singly bonded to a heteroatom substituent. the quantity is prepared in 3 elements facing sp3, sp2 and sp carbon associated with the heteroatoms. for every part cautious recognition has been given to varied good points reminiscent of substitution styles, ring results, pressure results, neighbouring performance, stereochemistry, and so on.

Comprehensive Medicinal Chemistry II, Volume 1

The 1st variation of accomplished Medicinal Chemistry used to be released in 1990 and used to be rather well acquired. accomplished Medicinal Chemistry II is way greater than an easy updating of the contents of the 1st version. thoroughly revised and elevated, this new version has been refocused to mirror the numerous advancements and adjustments over the last decade in genomics, proteomics, bioinformatics, combinatorial chemistry, high-throughput screening and pharmacology, and extra.

Terpene: Aromen, Düfte, Pharmaka, Pheromone

Einleitend werden die Bedeutung der Terpene, ihr als Isopren-Regel bekanntes Bauprinzip und ihre Biogenese skizziert. Es folgt eine nach Anzahl der Isopren-Einheiten und Grundskeletten geordnete Übersicht der bekanntesten Terpene, ihres Vorkommens in Pflanzen und anderen Organismen sowie ggf. ihrer biologischen und pharmakologischen Wirkungen.

Additional info for Annual Reports Medicinal Chemistry Volume 1

Sample text

42 (1964). A. M. Kasich. Curr. Therap. , 2 , 542 (1965). E. DePerrot, Psychiat. , 146,341 (1963b. a, D. Bente, M. P. Engelmeier, K. Heinrich, H. Hippius and W. Schmitt. , 14,538 (1964). J. Angst acd H. Kind, Schweiz. Med. , 2, 759 (1964). 0. H. Arnold, H. Bauer and K. Cmyral. Arzneimittel-Forsch.. 14. 510 (1964). H. Freeman, M. R . Otkem, M. W. Kristofferson and C. K. Gorby, Curr. Therap. R e s . , 1, 655 (1965) * I. W. Sletten, X. Pichardo and S. Gershon, Cum. Therap. , 1, 609 (1965). J. H. Biel, in Advances in Chemistry Series, No.

T h i s s i d e chain N-cyclopropylmethyl d e r i v a t i v e s i n has led t o p o t e n t a n t a g o n i s t s i n t h e morphine, morphinan and benzomorphan s e r i e s . I n t h e 6,14-endoethenothebaine s e r i e s when t h e C-alkanol s i d e chain i s isopropanol (XVIIIb) p o t e n t antagonism (35 x n a l o r p h i n e ) i s produced. =isoamyl (XVIIIc) t h e 1000 x compound behaves more l i k e a s t r o n g a n a l g e s i c (250 morphine). There were, however, some q u a l i t a t i v e d i f f e r e n c e s bet een XVIIIc and morphine.

Med. , 306 (1965). W. Wirth and R. Gosswald, Arch. int. Pharmacodyn.. 393 (1965). A. J. Glasky and L. N. Simon, Science, 702 (1966). N. Plotnikoff. Science, 703 (1966). E. N. Greenblatt and A. C. Osterberg. Toxicol. Appl. , 1, 566 (1965). '' ed. D. V. Siva Sankar, Art. 1, 1962, 1. Ann. N. Y. Acad. , 3. F. Downing, Quart. , X V I , 133 (1962). D. F. Downing, in Psychopharmacological Agents, Vol. I. ed. W. Gordon, Academic Press, New York-London. 1964. 555. A. Hoffer, Clin. Pharmacol. , 6 , 183 (1965).

Download PDF sample

Rated 5.00 of 5 – based on 4 votes